{"id":35058,"date":"2017-09-27T06:34:51","date_gmt":"2017-09-27T06:34:51","guid":{"rendered":"http:\/\/raed.academy\/?p=35058"},"modified":"2017-09-27T17:13:28","modified_gmt":"2017-09-27T17:13:28","slug":"una-molecula-contra-lalzheimer","status":"publish","type":"post","link":"https:\/\/raed.academy\/ca\/una-molecula-contra-lalzheimer\/","title":{"rendered":"Una mol\u00e8cula contra l&#8217;Alzheimer"},"content":{"rendered":"<h2>Francisco L\u00f3pez Mu\u00f1oz, acad\u00e8mic de la RAED, forma part de l&#8217;equip internacional que l&#8217;ha descoberta<\/h2>\n<p><a href=\"http:\/\/raed.academy\/ca\/academics\/dr-francisco-lopez-munoz\/\" target=\"_blank\" rel=\"noopener\"><strong>Francisco L\u00f3pez Mu\u00f1oz<\/strong><\/a>, acad\u00e8mic de n\u00famero de la <strong>Reial Acad\u00e8mia Europea de Doctors-Barcelona 1914<\/strong> (RAED), ha participat en un estudi multinacional que ha aconseguit identificar la mol\u00e8cula MBA354 com un agent neuroprotector, antioxidant i no t\u00f2xic que obre una nova via en la lluita contra l&#8217;Alzheimer. Publicat a l&#8217;edici\u00f3 internacional de la revista <strong>&#8220;Angewandte Chemie&#8221;<\/strong>, el treball confirma el potencial terap\u00e8utic d&#8217;aquesta mol\u00e8cula i obre noves i prometedores perspectives per a l&#8217;inici dels estudis precl\u00ednics per avaluar el seu potencial \u00fas en la ter\u00e0pia d&#8217;aquesta malaltia neurodegenerativa.<\/p>\n<p>Les dades de 2015 indiquen que 44 milions de persones es van veure afectades en el m\u00f3n per la malaltia d&#8217;Alzheimer, nombre que s&#8217;estima es duplicar\u00e0 en el 2030. Encara no s&#8217;ha trobat un f\u00e0rmac efica\u00e7 per a la seva ter\u00e0pia i el tractament, avui en dia, segueix sent limitat i pal\u00b7liatiu. En la recerca de noves vies per combatre-la, el disseny de mol\u00e8cules multipotents, capaces d&#8217;actuar simult\u00e0niament en diversos sistemes enzim\u00e0tics o receptors implicats en el progr\u00e9s i desenvolupament de la malaltia, \u00e9s una de les estrat\u00e8gies terap\u00e8utiques amb m\u00e9s expectatives.<\/p>\n<p>La mol\u00e8cula dissenyada per aquest equip internacional posseeix un car\u00e0cter tripotent, ja que \u00e9s capa\u00e7 d&#8217;inhibir les colinesterases i les monoaminooxidasas A \/ B i antagonitzar els receptors d&#8217;histamina H3R. A m\u00e9s, la mol\u00e8cula MBA354, que presenta un adequat perfil farmacol\u00f2gic in vitro i pot\u00e8ncies d&#8217;inhibici\u00f3 o interacci\u00f3 a nivell nanomolar, \u00e9s permeable a la barrera hematoencef\u00e0lica i presenta propietats antioxidants i neuroprotectores. Tamb\u00e9 ha mostrat un significatiu efecte procognitivo en un model in vivo de la malaltia d&#8217;Alzheimer, el que permetr\u00e0 ulteriors desenvolupaments encaminats a trobar un compost-lead per a la seva ter\u00e0pia.<\/p>\n<div id=\"attachment_35087\" style=\"width: 395px\" class=\"wp-caption alignright\"><img loading=\"lazy\" decoding=\"async\" aria-describedby=\"caption-attachment-35087\" class=\"wp-image-35087\" src=\"http:\/\/raed.academy\/wp-content\/uploads\/2017\/09\/Francisco-Lopez-mu\u00f1oz-alzheimer-w.jpg\" alt=\"Francisco Lopez Mu\u00f1oz - una mol\u00e8cula contra l'alzheimer\" width=\"385\" height=\"289\" \/><p id=\"caption-attachment-35087\" class=\"wp-caption-text\">Dr. Francisco L\u00f3pez Mu\u00f1oz<\/p><\/div>\n<p>Aquest equip multidisciplinari europeu est\u00e0 integrat per investigadors del <a href=\"http:\/\/www.csic.es\" target=\"_blank\" rel=\"noopener\"><strong>Consell Superior d&#8217;Investigacions Cient\u00edfiques<\/strong><\/a>, la <a href=\"http:\/\/www.ucjc.edu\" target=\"_blank\" rel=\"noopener\"><strong>Universitat Camilo Jos\u00e9 Cela<\/strong><\/a>, la <a href=\"http:\/\/www.ucm.es\" target=\"_blank\" rel=\"noopener\"><strong>Universitat Complutense de Madrid<\/strong><\/a>, la <a href=\"http:\/\/www.uah.es\" target=\"_blank\" rel=\"noopener\"><strong>Universitat d&#8217;Alcal\u00e1<\/strong><\/a>, l&#8217;<a href=\"http:\/\/www.madrid.org\/hospitaldelaprincesa\" target=\"_blank\" rel=\"noopener\"><strong>Hospital Universitari de la Princesa de Madrid<\/strong><\/a>, la <a href=\"http:\/\/www.uni-duesseldorf.de\" target=\"_blank\" rel=\"noopener\"><strong>Universitat Heinrich Heine de D\u00fcsseldorf<\/strong><\/a> (Alemanya) , la <a href=\"http:\/\/www.goethe-university-frankfurt.de\" target=\"_blank\" rel=\"noopener\"><strong>Universitat Goethe de Frankfurt<\/strong><\/a> (Alemanya), la <a href=\"http:\/\/www.st-andrews.ac.uk\" target=\"_blank\" rel=\"noopener\"><strong>Universitat de Saint Andrews<\/strong><\/a> (Regne Unit), la <a href=\"http:\/\/www.univ-fcomte.fr\" target=\"_blank\" rel=\"noopener\"><strong>Universitat de Franche-Comt\u00e9<\/strong><\/a> de Besan\u00e7on (Fran\u00e7a) i l&#8217;<a href=\"http:\/\/www.fnhk.cz\" target=\"_blank\" rel=\"noopener\"><strong>Hospital Universitari de Hradec Kr\u00e1lov\u00e9<\/strong><\/a> (Tx\u00e8quia).<\/p>\n<p>Sobre aquesta investigaci\u00f3 es va presentar una sol\u00b7licitud de patent el passat 23 d&#8217;agost a l&#8217;Oficina Espanyola de Patents i Marques amb el t\u00edtol &#8220;Nous compostos amb capacitat antioxidant que combinen la inhibici\u00f3 dels enzims monoaminoxidasas i colinesterases i la interacci\u00f3 amb el receptor d&#8217;histamina 3 , el seu procediment d&#8217;obtenci\u00f3 i composicions farmac\u00e8utiques que els contenen&#8221; a nom del Consell Superior d&#8217;Investigacions Cient\u00edfiques i la Universitat Camilo Jos\u00e9 Cela.<\/p>\n","protected":false},"excerpt":{"rendered":"<p>Francisco L\u00f3pez Mu\u00f1oz, acad\u00e8mic de la RAED, forma part de l&#8217;equip internacional que l&#8217;ha descoberta Francisco L\u00f3pez Mu\u00f1oz, acad\u00e8mic de n\u00famero de la Reial Acad\u00e8mia Europea de Doctors-Barcelona 1914 (RAED), ha participat en un estudi multinacional que ha aconseguit identificar la mol\u00e8cula MBA354 com un agent neuroprotector, antioxidant i no t\u00f2xic que obre una nova [&hellip;]<\/p>\n","protected":false},"author":12,"featured_media":0,"comment_status":"closed","ping_status":"closed","sticky":false,"template":"","format":"standard","meta":{"_et_pb_use_builder":"","_et_pb_old_content":"","_et_gb_content_width":"","footnotes":""},"categories":[72],"tags":[],"class_list":["post-35058","post","type-post","status-publish","format-standard","hentry","category-uncategorized-ca","et-doesnt-have-format-content","et_post_format-et-post-format-standard"],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v27.4 - 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